Basic Peptide Information

DICL ID
DICL_Pep_04379
Ion Channel
Sodium channel type 4 subunit alpha
Peptide Function
Inhibitor
Gene Name
Scn4a

Activity Data (nM)

IC50
61 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
DCLGFLWKCNPSNDKCCRPNLVCSRKDKWCKYQI
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Paurtx3; recombinant Paurtx-3 (rPaurtx-3)
Peptide Species
Paraphysa scrofa (Chilean copper tarantula) (Phrixotrichus auratus)
Peptide Name
Beta-theraphotoxin-Ps1a
CAS Number
Not available

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
22–25 °C
Test Method
Patch-clamping
Test Species
HEK293T cell (Homo sapiens embryonic kidney 293T cell)

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available